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-Structure paper
Title | Design of substituted bis-Tetrahydrofuran (bis-THF)-derived Potent HIV-1 Protease Inhibitors, Protein-ligand X-ray Structure, and Convenient Syntheses of bis-THF and Substituted bis-THF Ligands. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 2, Page 298-302, Year 2011 |
Publish date | Jan 10, 2011 (structure data deposition date) |
![]() | Ghosh, A.K. / Martyr, C.D. / Steffey, M. / Wang, Y.F. / Agniswamy, J. / Amano, M. / Weber, I.T. / Mitsuya, H. |
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Methods | X-ray diffraction |
Resolution | 1.4 Å |
Structure data | ![]() PDB-3qaa: |
Chemicals | ![]() ChemComp-G04: ![]() ChemComp-NA: ![]() ChemComp-CL: ![]() ChemComp-GOL: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / ![]() |