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-Structure paper
Title | Molecular Mechanism of Selectivity among G Protein-Coupled Receptor Kinase 2 Inhibitors. |
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Journal, issue, pages | Mol. Pharmacol., Vol. 80, Page 294-303, Year 2011 |
Publish date | Dec 1, 2010 (structure data deposition date) |
![]() | Thal, D.M. / Yeow, R.Y. / Schoenau, C. / Huber, J. / Tesmer, J.J. |
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Methods | X-ray diffraction |
Resolution | 2.48 - 2.67 Å |
Structure data | ![]() PDB-3psc: ![]() PDB-3pvu: ![]() PDB-3pvw: |
Chemicals | ![]() ChemComp-HOH: ![]() ChemComp-QRW: ![]() ChemComp-QRX: |
Source |
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![]() | TRANSFERASE/SIGNALING PROTEIN / Kinase / Serine/threonine-protein kinase / ATP-binding / Membrane / TRANSFERASE-SIGNALING PROTEIN complex / TRANSFERASE/SIGNALING PROTEIN/INHIBITOR / Transferase / Inhibitor / TRANSFERASE-SIGNALING PROTEIN-INHIBITOR complex |