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-Structure paper
Title | Non-oxime inhibitors of B-Raf(V600E) kinase. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 21, Page 1243-1247, Year 2011 |
Publish date | Nov 24, 2010 (structure data deposition date) |
Authors | Ren, L. / Wenglowsky, S. / Miknis, G. / Rast, B. / Buckmelter, A.J. / Ely, R.J. / Schlachter, S. / Laird, E.R. / Randolph, N. / Callejo, M. ...Ren, L. / Wenglowsky, S. / Miknis, G. / Rast, B. / Buckmelter, A.J. / Ely, R.J. / Schlachter, S. / Laird, E.R. / Randolph, N. / Callejo, M. / Martinson, M. / Galbraith, S. / Brandhuber, B.J. / Vigers, G. / Morales, T. / Voegtli, W.C. / Lyssikatos, J. |
External links | Bioorg. Med. Chem. Lett. / PubMed:21251822 |
Methods | X-ray diffraction |
Resolution | 2.9 - 3.7 Å |
Structure data | PDB-3ppj: PDB-3ppk: PDB-3prf: PDB-3pri: |
Chemicals | ChemComp-FOI: ChemComp-FNI: ChemComp-FP3: ChemComp-FP4: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / Protein kinase / ATP-competitive inhibitor / TRANSFERASE-TRANSFERASE INHIBITOR complex / B-Raf ATP-competitive inhibitor |