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-Structure paper
Title | Identification and development of novel inhibitors of Toxoplasma gondii enoyl reductase. |
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Journal, issue, pages | J. Med. Chem., Vol. 53, Page 6287-6300, Year 2010 |
Publish date | Jun 17, 2010 (structure data deposition date) |
Authors | Tipparaju, S.K. / Muench, S.P. / Mui, E.J. / Ruzheinikov, S.N. / Lu, J.Z. / Hutson, S.L. / Kirisits, M.J. / Prigge, S.T. / Roberts, C.W. / Henriquez, F.L. ...Tipparaju, S.K. / Muench, S.P. / Mui, E.J. / Ruzheinikov, S.N. / Lu, J.Z. / Hutson, S.L. / Kirisits, M.J. / Prigge, S.T. / Roberts, C.W. / Henriquez, F.L. / Kozikowski, A.P. / Rice, D.W. / McLeod, R.L. |
External links | J. Med. Chem. / PubMed:20698542 |
Methods | X-ray diffraction |
Resolution | 2.7 Å |
Structure data | PDB-3nj8: |
Chemicals | ChemComp-NAD: ChemComp-NJ8: ChemComp-HOH: |
Source |
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Keywords | OXIDOREDUCTASE / enoyl reductase / ENR triclosan / Rossmann NAD binding fold / NADH binding |