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-Structure paper
Title | Binding or bending: distinction of allosteric Abl kinase agonists from antagonists by an NMR-based conformational assay. |
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Journal, issue, pages | J. Am. Chem. Soc., Vol. 132, Page 7043-7048, Year 2010 |
Publish date | Apr 29, 2010 (structure data deposition date) |
Authors | Jahnke, W. / Grotzfeld, R.M. / Pelle, X. / Strauss, A. / Fendrich, G. / Cowan-Jacob, S.W. / Cotesta, S. / Fabbro, D. / Furet, P. / Mestan, J. / Marzinzik, A.L. |
External links | J. Am. Chem. Soc. / PubMed:20450175 |
Methods | X-ray diffraction |
Resolution | 1.8 - 1.95 Å |
Structure data | PDB-3ms9: PDB-3mss: |
Chemicals | ChemComp-STI: ChemComp-MS9: ChemComp-CL: ChemComp-HOH: ChemComp-MS7: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE REGULATOR / kinase / fragment-based screening / FBS / TRANSFERASE / TRANSFERASE-TRANSFERASE REGULATOR complex / TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE-TRANSFERASE INHIBITOR complex |