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-Structure paper
Title | Discovery of the Highly Potent PI3K/mTOR Dual Inhibitor PF-04979064 through Structure-Based Drug Design. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 4, Page 91-97, Year 2013 |
Publish date | Apr 16, 2010 (structure data deposition date) |
![]() | Cheng, H. / Li, C. / Bailey, S. / Baxi, S.M. / Goulet, L. / Guo, L. / Hoffman, J. / Jiang, Y. / Johnson, T.O. / Johnson, T.W. ...Cheng, H. / Li, C. / Bailey, S. / Baxi, S.M. / Goulet, L. / Guo, L. / Hoffman, J. / Jiang, Y. / Johnson, T.O. / Johnson, T.W. / Knighton, D.R. / Li, J. / Liu, K.K. / Liu, Z. / Marx, M.A. / Walls, M. / Wells, P.A. / Yin, M.J. / Zhu, J. / Zientek, M. |
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Methods | X-ray diffraction |
Resolution | 2.35 - 2.7 Å |
Structure data | ![]() PDB-3ml8: ![]() PDB-3ml9: ![]() PDB-4hvb: |
Chemicals | ![]() ChemComp-ML8: ![]() ChemComp-ML9: ![]() ChemComp-HOH: ![]() ChemComp-19P: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / phosphoinositide kinase / inhibition / TRANSFERASE / TRANSFERASE-TRANSFERASE INHIBITOR complex / Lipid kinase / kinase |