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| Title | Novel insights for dihydroorotate dehydrogenase class 1A inhibitors discovery. |
|---|---|
| Journal, issue, pages | Eur. J. Med. Chem., Vol. 45, Page 5899-5909, Year 2010 |
| Publish date | Apr 8, 2010 (structure data deposition date) |
Authors | Cheleski, J. / Rocha, J.R. / Pinheiro, M.P. / Wiggers, H.J. / da Silva, A.B. / Nonato, M.C. / Montanari, C.A. |
External links | Eur. J. Med. Chem. / PubMed:20965617 |
| Methods | X-ray diffraction |
| Resolution | 1.85 - 1.96 Å |
| Structure data | ![]() PDB-3mhu: ![]() PDB-3mjy: |
| Chemicals | ![]() ChemComp-FMN: ![]() ChemComp-EJZ: ![]() ChemComp-GOL: ![]() ChemComp-SO4: ![]() ChemComp-HOH: ![]() ChemComp-IJZ: |
| Source |
|
Keywords | OXIDOREDUCTASE / dihydroorotate dehydrogenase / pyrd |
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leishmania major (eukaryote)
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