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-Structure paper
Title | New potent dual inhibitors of CK2 and Pim kinases: discovery and structural insights. |
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Journal, issue, pages | Faseb J., Vol. 24, Page 3171-3185, Year 2010 |
Publish date | Mar 23, 2010 (structure data deposition date) |
![]() | Lopez-Ramos, M. / Prudent, R. / Moucadel, V. / Sautel, C.F. / Barette, C. / Lafanechere, L. / Mouawad, L. / Grierson, D. / Schmidt, F. / Florent, J.C. ...Lopez-Ramos, M. / Prudent, R. / Moucadel, V. / Sautel, C.F. / Barette, C. / Lafanechere, L. / Mouawad, L. / Grierson, D. / Schmidt, F. / Florent, J.C. / Filippakopoulos, P. / Bullock, A.N. / Knapp, S. / Reiser, J.B. / Cochet, C. |
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Methods | X-ray diffraction |
Resolution | 1.65 - 2.3 Å |
Structure data | ![]() PDB-3ma3: ![]() PDB-3mb6: ![]() PDB-3mb7: |
Chemicals | ![]() ChemComp-01I: ![]() ChemComp-HOH: ![]() ChemComp-SO4: ![]() ChemComp-14I: |
Source |
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![]() | TRANSFERASE / ONCOGENE / KINASE / SERINE-THREONINE / PIM1 / STRUCTURAL GENOMICS CONSORTIUM / SGC / ALTERNATIVE INITIATION / ATP-BINDING / MANGANESE / MEMBRANE / METAL-BINDING / NUCLEOTIDE-BINDING / NUCLEUS / PHOSPHOPROTEIN / PROTO-ONCOGENE / SERINE/THREONINE-PROTEIN KINASE / HOST-VIRUS INTERACTION / VIRAL IMMUNOEVASION / VIRION / VIRULENCE / Cell cycle / Cell membrane / kinases / difurane / inhibitor / CK2 |