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-Structure paper
Title | Structure and activity relationships of tartrate-based TACE inhibitors. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 20, Page 4812-4815, Year 2010 |
Publish date | Jan 21, 2010 (structure data deposition date) |
Authors | Li, D. / Popovici-Muller, J. / Belanger, D.B. / Caldwell, J. / Dai, C. / David, M. / Girijavallabhan, V.M. / Lavey, B.J. / Lee, J.F. / Liu, Z. ...Li, D. / Popovici-Muller, J. / Belanger, D.B. / Caldwell, J. / Dai, C. / David, M. / Girijavallabhan, V.M. / Lavey, B.J. / Lee, J.F. / Liu, Z. / Mazzola, R. / Rizvi, R. / Rosner, K.E. / Shankar, B. / Spitler, J. / Ting, P.C. / Vaccaro, H. / Yu, W. / Zhou, G. / Zhu, Z. / Niu, X. / Sun, J. / Guo, Z. / Orth, P. / Chen, S. / Kozlowski, J.A. / Lundell, D.J. / Madison, V. / McKittrick, B. / Piwinski, J.J. / Shih, N.Y. / Shipps, G.W. / Siddiqui, M.A. / Strickland, C.O. |
External links | Bioorg. Med. Chem. Lett. / PubMed:20638281 |
Methods | X-ray diffraction |
Resolution | 1.9 Å |
Structure data | PDB-3lgp: |
Chemicals | ChemComp-ZN: ChemComp-50X: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / GLYCOPROTEIN / MEMBRANE / METAL-BINDING / METALLOPROTEASE / NOTCH SIGNALING PATHWAY / PHOSPHOPROTEIN / PROTEASE / TRANSMEMBRANE / ZYMOGEN / Cleavage on pair of basic residues / Disulfide bond / SH3-binding |