+Search query
-Structure paper
Title | Potent and Selective Inhibition of Polycythemia by the Quinoxaline JAK2 Inhibitor NVP-BSK805 |
---|---|
Journal, issue, pages | Mol. Cancer Ther., Vol. 9, Page 1945-1955, Year 2010 |
Publish date | Nov 19, 2009 (structure data deposition date) |
![]() | Baffert, F. / Regnier, C.H. / De Pover, A. / Pissot-Soldermann, C. / Tavares, G.A. / Blasco, F. / Brueggen, J. / Chene, P. / Drueckes, P. / Erdmann, D. ...Baffert, F. / Regnier, C.H. / De Pover, A. / Pissot-Soldermann, C. / Tavares, G.A. / Blasco, F. / Brueggen, J. / Chene, P. / Drueckes, P. / Erdmann, D. / Furet, P. / Gerspacher, M. / Lang, M. / Ledieu, D. / Nolan, L. / Ruetz, S. / Trappe, J. / Vangrevelinghe, E. / Wartmann, M. / Wyder, L. / Hofmann, F. / Radimerski, T. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.8 Å |
Structure data | ![]() PDB-3krr: |
Chemicals | ![]() ChemComp-DQX: ![]() ChemComp-HOH: |
Source |
|
![]() | TRANSFERASE / Small molecule inhibitor / ATP site kinase inhibitor / ATP-binding / Disease mutation / Kinase / Membrane / Nucleotide-binding / Phosphoprotein / Proto-oncogene / SH2 domain / Tyrosine-protein kinase |