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-Structure paper
Title | Design and Synthesis of Potent and Selective BACE-1 Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 53, Page 1458-1464, Year 2010 |
Publish date | Sep 4, 2009 (structure data deposition date) |
![]() | Bjorklund, C. / Oscarson, S. / Benkestock, K. / Borkakoti, N. / Jansson, K. / Lindberg, J. / Vrang, L. / Hallberg, A. / Rosenquist, A. / Samuelsson, B. |
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Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | ![]() PDB-3ixj: |
Chemicals | ![]() ChemComp-586: ![]() ChemComp-SO4: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / BACE / BETA SECRETASE-1 / INHIBITOR / ALTERNATIVE SPLICING / ASPARTYL PROTEASE / GLYCOPROTEIN / HYDROLASE / MEMBRANE / PROTEASE / TRANSMEMBRANE / ZYMOGEN / Disulfide bond / Polymorphism / HYDROLASE-HYDROLASE INHIBITOR COMPLEX |