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-Structure paper
Title | Novel mutant-selective EGFR kinase inhibitors against EGFR T790M. |
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Journal, issue, pages | Nature, Vol. 462, Page 1070-1074, Year 2009 |
Publish date | Aug 5, 2009 (structure data deposition date) |
Authors | Zhou, W. / Ercan, D. / Chen, L. / Yun, C.H. / Li, D. / Capelletti, M. / Cortot, A.B. / Chirieac, L. / Iacob, R.E. / Padera, R. ...Zhou, W. / Ercan, D. / Chen, L. / Yun, C.H. / Li, D. / Capelletti, M. / Cortot, A.B. / Chirieac, L. / Iacob, R.E. / Padera, R. / Engen, J.R. / Wong, K.K. / Eck, M.J. / Gray, N.S. / Janne, P.A. |
External links | Nature / PubMed:20033049 |
Methods | X-ray diffraction |
Resolution | 2.9 Å |
Structure data | PDB-3ika: |
Chemicals | ChemComp-0UN: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / EGFR / T790M / WZ4002 / WZ-4002 / Alternative splicing / ATP-binding / Cell membrane / Disease mutation / Disulfide bond / Glycoprotein / Isopeptide bond / Kinase / Membrane / Nucleotide-binding / Phosphoprotein / Polymorphism / Receptor / Secreted / Transmembrane / Tumor suppressor / Tyrosine-protein kinase / Ubl conjugation |