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-Structure paper
Title | Fluorophore labeling of the glycine-rich loop as a method of identifying inhibitors that bind to active and inactive kinase conformations. |
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Journal, issue, pages | J. Am. Chem. Soc., Vol. 132, Page 4152-4160, Year 2010 |
Publish date | Jun 13, 2009 (structure data deposition date) |
![]() | Simard, J.R. / Getlik, M. / Grutter, C. / Schneider, R. / Wulfert, S. / Rauh, D. |
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Methods | X-ray diffraction |
Resolution | 1.8 - 2.35 Å |
Structure data | ![]() PDB-3hub: ![]() PDB-3huc: ![]() PDB-3l8s: |
Chemicals | ![]() ChemComp-BOG: ![]() ChemComp-469: ![]() ChemComp-HOH: ![]() ChemComp-G97: ![]() ChemComp-MES: ![]() ChemComp-BFF: |
Source |
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![]() | TRANSFERASE / DFG-in / Glycine-Rich Loop / Scios-469 / Alternative splicing / ATP-binding / Cytoplasm / Kinase / Nucleotide-binding / Nucleus / Phosphoprotein / Polymorphism / Serine/threonine-protein kinase / DFG-out / CP-547632 |