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Structure paper

TitleAminopiperidine-fused imidazoles as dipeptidyl peptidase-IV inhibitors
Journal, issue, pagesBioorg. Med. Chem. Lett., Vol. 19, Page 4097-4101, Year 2009
Publish dateMay 1, 2009 (structure data deposition date)
AuthorsEdmondson, S.D. / Mastracchio, A. / Cox, J.M. / Eiermann, G.J. / He, H. / Lyons, K.A. / Patel, R.A. / Patel, S.B. / Petrov, A. / Scapin, G. ...Edmondson, S.D. / Mastracchio, A. / Cox, J.M. / Eiermann, G.J. / He, H. / Lyons, K.A. / Patel, R.A. / Patel, S.B. / Petrov, A. / Scapin, G. / Wu, J.K. / Xu, S. / Zhu, B. / Thornberry, N.A. / Roy, R.S. / Weber, A.E.
External linksBioorg. Med. Chem. Lett. / PubMed:19539471
MethodsX-ray diffraction
Resolution2 - 2.1 Å
Structure data

PDB-3hab:
The structure of DPP4 in complex with piperidine fused benzimidazole 25
Method: X-RAY DIFFRACTION / Resolution: 2.1 Å

PDB-3hac:
The structure of DPP-4 in complex with piperidine fused imidazopyridine 34
Method: X-RAY DIFFRACTION / Resolution: 2 Å

Chemicals

ChemComp-NAG:
2-acetamido-2-deoxy-beta-D-glucopyranose

ChemComp-NA:
Unknown entry

ChemComp-677:
(2R,3R)-7-(methylsulfonyl)-3-(2,4,5-trifluorophenyl)-1,2,3,4-tetrahydropyrido[1,2-a]benzimidazol-2-amine

ChemComp-HOH:
WATER

ChemComp-361:
(7R,8R)-8-(2,4,5-trifluorophenyl)-6,7,8,9-tetrahydroimidazo[1,2-a:4,5-c']dipyridin-7-amine

Source
  • homo sapiens (human)
KeywordsHYDROLASE/HYDROLASE INHIBITOR / ALPHA/BETA / BETA-PROPELLER / DIMER / HYDROLASE / DIABETES / Aminopeptidase / Cell membrane / Disulfide bond / Glycoprotein / Membrane / Protease / Secreted / Serine protease / Signal-anchor / Transmembrane / HYDROLASE-HYDROLASE INHIBITOR COMPLEX

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