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TitleN-aryl-oxazolidin-2-imine muscle selective androgen receptor modulators enhance potency through pharmacophore reorientation.
Journal, issue, pagesJ. Med. Chem., Vol. 52, Page 2794-2798, Year 2009
Publish dateJan 29, 2009 (structure data deposition date)
AuthorsNirschl, A.A. / Zou, Y. / Krystek, S.R. / Sutton, J.C. / Simpkins, L.M. / Lupisella, J.A. / Kuhns, J.E. / Seethala, R. / Golla, R. / Sleph, P.G. ...Nirschl, A.A. / Zou, Y. / Krystek, S.R. / Sutton, J.C. / Simpkins, L.M. / Lupisella, J.A. / Kuhns, J.E. / Seethala, R. / Golla, R. / Sleph, P.G. / Beehler, B.C. / Grover, G.J. / Egan, D. / Fura, A. / Vyas, V.P. / Li, Y.X. / Sack, J.S. / Kish, K.F. / An, Y. / Bryson, J.A. / Gougoutas, J.Z. / DiMarco, J. / Zahler, R. / Ostrowski, J. / Hamann, L.G.
External linksJ. Med. Chem. / PubMed:19351168
MethodsX-ray diffraction
Resolution1.95 Å
Structure data

PDB-3g0w:
Crystal structure of the rat androgen receptor ligand binding domain complex with an n-aryl-oxazolidin 2-imine inhibitor
Method: X-RAY DIFFRACTION / Resolution: 1.95 Å

Chemicals

ChemComp-LGB:
2-chloro-4-{[(1R,3Z,7S,7aS)-7-hydroxy-1-(trifluoromethyl)tetrahydro-1H-pyrrolo[1,2-c][1,3]oxazol-3-ylidene]amino}-3-met

ChemComp-HOH:
WATER

Source
  • rattus norvegicus (Norway rat)
KeywordsHORMONE / ANDROGEN RECEPTOR / STEROID RECEPTOR / NUCLEAR RECEPTOR / TRANSCRIPTION REGULATION / LIGAND-BINDING DOMAIN / Disease mutation / DNA-binding / Lipid-binding / Metal-binding / Nucleus / Phosphoprotein / Receptor / Steroid-binding / Transcription / Ubl conjugation / Zinc / Zinc-finger / HORMONE-GROWTH FACTOR COMPLEX

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