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-Structure paper
Title | Designed inhibitors of insulin-degrading enzyme regulate the catabolism and activity of insulin. |
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Journal, issue, pages | Plos One, Vol. 5, Page e10504-e10504, Year 2010 |
Publish date | Aug 11, 2008 (structure data deposition date) |
![]() | Leissring, M.A. / Malito, E. / Hedouin, S. / Reinstatler, L. / Sahara, T. / Abdul-Hay, S.O. / Choudhry, S. / Maharvi, G.M. / Fauq, A.H. / Huzarska, M. ...Leissring, M.A. / Malito, E. / Hedouin, S. / Reinstatler, L. / Sahara, T. / Abdul-Hay, S.O. / Choudhry, S. / Maharvi, G.M. / Fauq, A.H. / Huzarska, M. / May, P.S. / Choi, S. / Logan, T.P. / Turk, B.E. / Cantley, L.C. / Manolopoulou, M. / Tang, W.J. / Stein, R.L. / Cuny, G.D. / Selkoe, D.J. |
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Methods | X-ray diffraction |
Resolution | 2.6 Å |
Structure data | ![]() PDB-3e4a: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-QIX: ![]() ChemComp-DIO: ![]() ChemComp-ACY: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE / INSULIN / HYDROXAMATE / INSULIN DEGRADING ENZYME / Metal-binding / Metalloprotease / Protease |