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-Structure paper
Title | Discovery of a novel class of potent human deoxyuridine triphosphatase inhibitors remarkably enhancing the antitumor activity of thymidylate synthase inhibitors |
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Journal, issue, pages | J. Med. Chem., Vol. 55, Page 2970-2980, Year 2012 |
Publish date | Dec 3, 2010 (structure data deposition date) |
![]() | Miyahara, S. / Miyakoshi, H. / Yokogawa, T. / Chong, K.T. / Taguchi, J. / Muto, T. / Endoh, K. / Yano, W. / Wakasa, T. / Ueno, H. ...Miyahara, S. / Miyakoshi, H. / Yokogawa, T. / Chong, K.T. / Taguchi, J. / Muto, T. / Endoh, K. / Yano, W. / Wakasa, T. / Ueno, H. / Takao, Y. / Fujioka, A. / Hashimoto, A. / Itou, K. / Yamamura, K. / Nomura, M. / Nagasawa, H. / Shuto, S. / Fukuoka, M. |
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Methods | X-ray diffraction |
Resolution | 1.8 Å |
Structure data | ![]() PDB-3arn: |
Chemicals | ![]() ChemComp-MSJ: ![]() ChemComp-MG: ![]() ChemComp-HOH: |
Source |
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![]() | Hydrolase/Hydrolase inhibitor / Hydrolase / Hydrolase-Hydrolase inhibitor complex |