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-Structure paper
Title | Development of a novel selective inhibitor of the Down syndrome-related kinase Dyrk1A |
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Journal, issue, pages | Nat Commun, Vol. 1, Page 1-9, Year 2010 |
Publish date | Sep 6, 2010 (structure data deposition date) |
![]() | Ogawa, Y. / Nonaka, Y. / Goto, T. / Ohnishi, E. / Hiramatsu, T. / Kii, I. / Yoshida, M. / Ikura, T. / Onogi, H. / Shibuya, H. ...Ogawa, Y. / Nonaka, Y. / Goto, T. / Ohnishi, E. / Hiramatsu, T. / Kii, I. / Yoshida, M. / Ikura, T. / Onogi, H. / Shibuya, H. / Hosoya, T. / Ito, N. / Hagiwara, M. |
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Methods | X-ray diffraction |
Resolution | 2.6 Å |
Structure data | ![]() PDB-3anq: ![]() PDB-3anr: |
Chemicals | ![]() ChemComp-EHB: ![]() ChemComp-HOH: ![]() ChemComp-HRM: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / protein kinase / TRANSFERASE / TRANSFERASE-TRANSFERASE INHIBITOR complex |