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Structure paper

TitleDiscovery of novel 3,6-disubstituted 2-pyridinecarboxamide derivatives as GK activators
Journal, issue, pagesBioorg. Med. Chem. Lett., Vol. 19, Page 2718-2721, Year 2009
Publish dateMar 19, 2009 (structure data deposition date)
AuthorsMitsuya, M. / Kamata, K. / Bamba, M. / Watanabe, H. / Sasaki, Y. / Sasaki, K. / Ohyama, S. / Hosaka, H. / Nagata, Y. / Eiki, J. / Nishimura, T.
External linksBioorg. Med. Chem. Lett. / PubMed:19362831
MethodsX-ray diffraction
Resolution2.2 - 2.52 Å
Structure data

PDB-3a0i:
Human glucokinase in complex with a synthetic activator
Method: X-RAY DIFFRACTION / Resolution: 2.2 Å

PDB-3goi:
Human glucokinase in complex with a synthetic activator
Method: X-RAY DIFFRACTION / Resolution: 2.52 Å

Chemicals

ChemComp-GLC:
alpha-D-glucopyranose

ChemComp-AJI:
3-[(4-fluorophenyl)sulfanyl]-N-(4-methyl-1,3-thiazol-2-yl)-6-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]pyridine-2-carboxamide

ChemComp-NA:
Unknown entry

ChemComp-HOH:
WATER

ChemComp-LOI:
2-(methylamino)-N-(4-methyl-1,3-thiazol-2-yl)-5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]benzamide

Source
  • homo sapiens (human)
KeywordsTRANSFERASE / Glucokinase / Diabetes / Activator / Alternative splicing / ATP-binding / Diabetes mellitus / Disease mutation / Glycolysis / Kinase / Nucleotide-binding / Polymorphism / allosteric activator

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