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-Structure paper
Title | Design and synthesis of peptidomimetic factor VIIa inhibitors |
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Journal, issue, pages | Chem. Pharm. Bull., Vol. 58, Page 38-44, Year 2010 |
Publish date | Feb 25, 2009 (structure data deposition date) |
Authors | Shiraishi, T. / Kadono, S. / Haramura, M. / Kodama, H. / Ono, Y. / Iikura, H. / Esaki, T. / Koga, T. / Hattori, K. / Watanabe, Y. ...Shiraishi, T. / Kadono, S. / Haramura, M. / Kodama, H. / Ono, Y. / Iikura, H. / Esaki, T. / Koga, T. / Hattori, K. / Watanabe, Y. / Sakamoto, A. / Yoshihashi, K. / Kitazawa, T. / Esaki, K. / Ohta, M. / Sato, H. / Kozono, T. |
External links | Chem. Pharm. Bull. / PubMed:20045964 |
Methods | X-ray diffraction |
Resolution | 2.5 Å |
Structure data | PDB-2zzu: |
Chemicals | ChemComp-BGC: ChemComp-FUC: ChemComp-CA: ChemComp-359: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE/BLOOD CLOTTING / SERINE PROTEASE / BLOOD COAGULATION / CLEAVAGE ON PAIR OF BASIC RESIDUES / DISEASE MUTATION / EGF-LIKE DOMAIN / GAMMA-CARBOXYGLUTAMIC ACID / GLYCOPROTEIN / HYDROLASE / HYDROXYLATION / PROTEASE / ZYMOGEN / LIPOPROTEIN / MEMBRANE / PALMITATE / TRANSMEMBRANE / HYDROLASE-BLOOD CLOTTING COMPLEX / SECRETED |