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| Title | Crystal structure of the Ca2+/calmodulin-dependent protein kinase kinase in complex with the inhibitor STO-609 |
|---|---|
| Journal, issue, pages | J. Biol. Chem., Vol. 286, Page 22570-22579, Year 2011 |
| Publish date | Oct 31, 2008 (structure data deposition date) |
Authors | Kukimoto-Niino, M. / Yoshikawa, S. / Takagi, T. / Ohsawa, N. / Tomabechi, Y. / Terada, T. / Shirouzu, M. / Suzuki, A. / Lee, S. / Yamauchi, T. ...Kukimoto-Niino, M. / Yoshikawa, S. / Takagi, T. / Ohsawa, N. / Tomabechi, Y. / Terada, T. / Shirouzu, M. / Suzuki, A. / Lee, S. / Yamauchi, T. / Okada-Iwabu, M. / Iwabu, M. / Kadowaki, T. / Minokoshi, Y. / Yokoyama, S. |
External links | J. Biol. Chem. / PubMed:21504895 |
| Methods | X-ray diffraction |
| Resolution | 2.4 Å |
| Structure data | ![]() PDB-2zv2: |
| Chemicals | ![]() ChemComp-609: ![]() ChemComp-HOH: |
| Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / calcium/calmodulin-dependent protein kinase kinase 2 / beta / STO-609 / CaMKK2 / E.C.2.7.11.17 / Phosphorylation / AMPKK / metabolism / ATP-binding / kinase / Calmodulin-binding / Nucleotide-binding / Phosphoprotein / Serine/threonine-protein kinase / Transferase / Structural Genomics / NPPSFA / National Project on Protein Structural and Functional Analyses / RIKEN Structural Genomics/Proteomics Initiative / RSGI / TRANSFERASE-TRANSFERASE INHIBITOR complex |
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