+Search query
-Structure paper
Title | Halogen Bonding at the Active Sites of Human Cathepsin L and Mek1 Kinase: Efficient Interactions in Different Environments. |
---|---|
Journal, issue, pages | Chemmedchem, Vol. 6, Page 2048-, Year 2011 |
Publish date | May 18, 2011 (structure data deposition date) |
Authors | Hardegger, L.A. / Kuhn, B. / Spinnler, B. / Anselm, L. / Ecabert, R. / Stihle, M. / Gsell, B. / Thoma, R. / Diez, J. / Benz, J.M. ...Hardegger, L.A. / Kuhn, B. / Spinnler, B. / Anselm, L. / Ecabert, R. / Stihle, M. / Gsell, B. / Thoma, R. / Diez, J. / Benz, J.M. / Plancher, J. / Hartmann, G. / Isshiki, Y. / Morikami, K. / Shimma, N. / Haap, W. / Banner, D.W. / Diederich, F. |
External links | Chemmedchem / PubMed:21898833 |
Methods | X-ray diffraction |
Resolution | 1.14 - 1.4 Å |
Structure data | PDB-2yj2: PDB-2yj8: PDB-2yj9: PDB-2yjb: PDB-2yjc: |
Chemicals | ChemComp-YJ2: ChemComp-GOL: ChemComp-HOH: ChemComp-YJ8: ChemComp-YJ9: ChemComp-424: |
Source |
|
Keywords | HYDROLASE / DRUG DESIGN / THIOL PROTEASE / INHIBITOR |