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-Structure paper
Title | Discovery and Characterization of Small Molecule Inhibitors of the Bet Family Bromodomains. |
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Journal, issue, pages | J. Med. Chem., Vol. 54, Page 3827-, Year 2011 |
Publish date | Mar 24, 2011 (structure data deposition date) |
![]() | Chung, C.W. / Coste, H. / White, J.H. / Mirguet, O. / Wilde, J. / Gosmini, R.L. / Delves, C. / Magny, S.M. / Woodward, R. / Hughes, S.A. ...Chung, C.W. / Coste, H. / White, J.H. / Mirguet, O. / Wilde, J. / Gosmini, R.L. / Delves, C. / Magny, S.M. / Woodward, R. / Hughes, S.A. / Boursier, E.V. / Flynn, H. / Bouillot, A.M. / Bamborough, P. / Brusq, J.M. / Gellibert, F.J. / Jones, E.J. / Riou, A.M. / Homes, P. / Martin, S.L. / Uings, I.J. / Toum, J. / Clement, C.A. / Boullay, A.B. / Grimley, R.L. / Blandel, F.M. / Prinjha, R.K. / Lee, K. / Kirilovsky, J. / Nicodeme, E. |
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Methods | X-ray diffraction |
Resolution | 1.65 - 2.3 Å |
Structure data | ![]() PDB-2ydw: ![]() PDB-2yek: ![]() PDB-2yel: ![]() PDB-2yem: |
Chemicals | ![]() ChemComp-WSH: ![]() ChemComp-SO4: ![]() ChemComp-HOH: ![]() ChemComp-EAM: ![]() ChemComp-EDO: |
Source |
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![]() | NUCLEAR PROTEIN / HISTONE / EPIGENETIC READER / SIGNALING PROTEIN |