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-Structure paper
Title | Thieno[3,2-C]Pyrazoles: A Novel Class of Aurora Inhibitors with Favorable Antitumor Activity. |
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Journal, issue, pages | Bioorg. Med. Chem., Vol. 18, Page 7113-, Year 2010 |
Publish date | Sep 22, 2010 (structure data deposition date) |
Authors | Bindi, S. / Fancelli, D. / Alli, C. / Berta, D. / Bertrand, J.A. / Cameron, A.D. / Cappella, P. / Carpinelli, P. / Cervi, G. / Croci, V. ...Bindi, S. / Fancelli, D. / Alli, C. / Berta, D. / Bertrand, J.A. / Cameron, A.D. / Cappella, P. / Carpinelli, P. / Cervi, G. / Croci, V. / D'Anello, M. / Forte, B. / Laura Giorgini, M. / Marsiglio, A. / Moll, J. / Pesenti, E. / Pittala, V. / Pulici, M. / Riccardi-Sirtori, F. / Roletto, F. / Soncini, C. / Storici, P. / Varasi, M. / Volpi, D. / Zugnoni, P. / Vianello, P. |
External links | Bioorg. Med. Chem. / PubMed:20817473 |
Methods | X-ray diffraction |
Resolution | 2.9 Å |
Structure data | PDB-2xru: |
Chemicals | ChemComp-400: |
Source |
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Keywords | TRANSFERASE / NUCLEOTIDE-BINDING / KINASE / CELL CYCLE |