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-Structure paper
Title | Toward the Rational Design of P53-Stabilizing Drugs: Probing the Surface of the Oncogenic Y220C Mutant. |
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Journal, issue, pages | Chem. Biol., Vol. 17, Page 46-, Year 2010 |
Publish date | Dec 17, 2009 (structure data deposition date) |
![]() | Basse, N. / Kaar, J.L. / Settanni, G. / Joerger, A.C. / Rutherford, T.J. / Fersht, A.R. |
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Methods | X-ray diffraction |
Resolution | 1.6 - 2.1 Å |
Structure data | ![]() PDB-2x0u: ![]() PDB-2x0v: ![]() PDB-2x0w: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-X0U: ![]() ChemComp-HOH: ![]() ChemComp-X0V: ![]() ChemComp-X0W: |
Source |
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![]() | CELL CYCLE / ACTIVATOR / TRANSCRIPTION REGULATION / TRANSCRIPTION FACTOR / LI-FRAUMENI DRUG DISCOVERY / SURFACE CREVICE / TUMOR SUPPRESSOR / PROTEIN STABILIZATION / TRANSCRIPTION / METAL BINDING / CANCER / APOPTOSIS / HOST-VIRUS INTERACTION / LI-FRAUMENI SYNDROME / DRUG DISCOVERY |