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TitleIdentification of Potent Pyrazolo[4,3-H]Quinazoline-3-Carboxamides as Multi-Cyclin-Dependent Kinase Inhibitors.
Journal, issue, pagesJ. Med. Chem., Vol. 53, Page 2171-, Year 2010
Publish dateNov 10, 2009 (structure data deposition date)
AuthorsTraquandi, G. / Ciomei, M. / Ballinari, D. / Casale, E. / Colombo, N. / Croci, V. / Fiorentini, F. / Isacchi, A. / Longo, A. / Mercurio, C. ...Traquandi, G. / Ciomei, M. / Ballinari, D. / Casale, E. / Colombo, N. / Croci, V. / Fiorentini, F. / Isacchi, A. / Longo, A. / Mercurio, C. / Panzeri, A. / Pastori, W. / Pevarello, P. / Volpi, D. / Roussel, P. / Vulpetti, A. / Brasca, M.G.
External linksJ. Med. Chem. / PubMed:20141146
MethodsX-ray diffraction
Resolution2.6 Å
Structure data

PDB-2wxv:
Structure of CDK2-CYCLIN A with a Pyrazolo(4,3-h) quinazoline-3- carboxamide inhibitor
Method: X-RAY DIFFRACTION / Resolution: 2.6 Å

Chemicals

ChemComp-WXV:
N,1-DIMETHYL-8-{[1-(METHYLSULFONYL)PIPERIDIN-4-YL]AMINO}-1H-PYRAZOLO[4,3-H]QUINAZOLINE-3-CARBOXAMIDE

ChemComp-SO4:
SULFATE ION

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsTRANSFERASE / NUCLEOTIDE-BINDING / SERINE/THREONINE-PROTEIN KINASE / CELL CYCLE / KINASE / CYCLIN

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