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| Title | Cellular Inhibition of Chk2 Kinase and Potentiation of Camptothecins and Radiation by the Novel Chk2 Inhibitor Pv1019. |
|---|---|
| Journal, issue, pages | J. Pharmacol. Exp. Ther., Vol. 331, Page 816-, Year 2009 |
| Publish date | Jan 6, 2009 (structure data deposition date) |
Authors | Jobson, A.G. / Lountos, G.T. / Lorenzi, P.L. / Llamas, J. / Connelly, J. / Cerna, D. / Tropea, J.E. / Onda, A. / Zoppoli, G. / Kondapaka, S. ...Jobson, A.G. / Lountos, G.T. / Lorenzi, P.L. / Llamas, J. / Connelly, J. / Cerna, D. / Tropea, J.E. / Onda, A. / Zoppoli, G. / Kondapaka, S. / Zhang, G. / Caplen, N.J. / Cardellina, J.H. / Yoo, S.S. / Monks, A. / Self, C. / Waugh, D.S. / Shoemaker, R.H. / Pommier, Y. |
External links | J. Pharmacol. Exp. Ther. / PubMed:19741151 |
| Methods | X-ray diffraction |
| Resolution | 2.07 Å |
| Structure data | ![]() PDB-2w7x: |
| Chemicals | ![]() ChemComp-D1A: ![]() ChemComp-MG: ![]() ChemComp-NO3: ![]() ChemComp-EDO: ![]() ChemComp-HOH: |
| Source |
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Keywords | TRANSFERASE / CO-CRYSTAL STRUCTURE / KINASE / NUCLEUS / MAGNESIUM / CELL CYCLE / ATP-BINDING / LI-FRAUMENI SYNDROME / SERINE/THREONINE-PROTEIN KINASE / DISEASE MUTATION / NUCLEOTIDE-BINDING / POTENTIATION / METAL-BINDING / PROTO-ONCOGENE / PHOSPHOPROTEIN / CHK2 INHIBITOR |
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homo sapiens (human)
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