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-Structure paper
Title | Structural Basis for Ligand Promiscuity in Cytochrome P450 3A4 |
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Journal, issue, pages | Proc. Natl. Acad. Sci. USA, Vol. 103, Page 13682-, Year 2006 |
Publish date | Aug 2, 2006 (structure data deposition date) |
Authors | Ekroos, M. / Sjogren, T. |
External links | Proc. Natl. Acad. Sci. USA / PubMed:16954191 |
Methods | X-ray diffraction |
Resolution | 2.75 - 2.8 Å |
Structure data | PDB-2j0d: PDB-2v0m: |
Chemicals | ChemComp-HEM: ChemComp-ERY: ChemComp-HOH: ChemComp-KLN: |
Source |
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Keywords | OXIDOREDUCTASE / POLYMORPHISM / ERYTHROMYCIN / MONOOXYGENASE / METAL-BINDING / TRANSMEMBRANE / ENDOPLASMIC RETICULUM / DRUG METABOLIZING ENZYME / P450 / NADP / IRON / HEME / CYP3A4 / MEMBRANE / MICROSOME / KETOCONAZOL |