+Search query
-Structure paper
Title | Distinct Structural Mechanisms for Inhibition of Pyruvate Dehydrogenase Kinase Isoforms by AZD7545, Dichloroacetate, and Radicicol. |
---|---|
Journal, issue, pages | Structure, Vol. 15, Page 992-1004, Year 2007 |
Publish date | Jun 10, 2007 (structure data deposition date) |
![]() | Kato, M. / Li, J. / Chuang, J.L. / Chuang, D.T. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.9 - 2.6 Å |
Structure data | ![]() PDB-2q8f: ![]() PDB-2q8g: ![]() PDB-2q8h: ![]() PDB-2q8i: |
Chemicals | ![]() ChemComp-K: ![]() ChemComp-HOH: ![]() ChemComp-AZX: ![]() ChemComp-TF4: ![]() ChemComp-RDC: ![]() ChemComp-GOL: ![]() ChemComp-RED: |
Source |
|
![]() | TRANSFERASE / GHKL ATPase/kinase family / pyruvate dehydrogenase complex / mitochondrial kinase / glucose-lowering drug AZD7545 / dichroloacetate / radicicol |