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-Structure paper
Title | Flipped Out: Structure-Guided Design of Selective Pyrazolylpyrrole ERK Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 50, Page 1280-1287, Year 2007 |
Publish date | Jan 12, 2007 (structure data deposition date) |
Authors | Aronov, A.M. / Baker, C. / Bemis, G.W. / Cao, J. / Chen, G. / Ford, P.J. / Germann, U.A. / Green, J. / Hale, M.R. / Jacobs, M. ...Aronov, A.M. / Baker, C. / Bemis, G.W. / Cao, J. / Chen, G. / Ford, P.J. / Germann, U.A. / Green, J. / Hale, M.R. / Jacobs, M. / Janetka, J.W. / Maltais, F. / Martinez-Botella, G. / Namchuk, M.N. / Straub, J. / Tang, Q. / Xie, X. |
External links | J. Med. Chem. / PubMed:17300186 |
Methods | X-ray diffraction |
Resolution | 2 - 2.6 Å |
Structure data | PDB-2ojg: PDB-2oji: PDB-2ojj: PDB-2ok1: |
Chemicals | ChemComp-SO4: ChemComp-19A: ChemComp-HOH: ChemComp-33A: ChemComp-82A: |
Source |
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Keywords | TRANSFERASE / kinase inhibitor |