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TitleDiscovery of non-covalent dipeptidyl peptidase IV inhibitors which induce a conformational change in the active site.
Journal, issue, pagesBioorg. Med. Chem. Lett., Vol. 17, Page 1765-1768, Year 2007
Publish dateJan 9, 2007 (structure data deposition date)
AuthorsSheehan, S.M. / Mest, H.J. / Watson, B.M. / Klimkowski, V.J. / Timm, D.E. / Cauvin, A. / Parsons, S.H. / Shi, Q. / Canada, E.J. / Wiley, M.R. ...Sheehan, S.M. / Mest, H.J. / Watson, B.M. / Klimkowski, V.J. / Timm, D.E. / Cauvin, A. / Parsons, S.H. / Shi, Q. / Canada, E.J. / Wiley, M.R. / Ruehter, G. / Evers, B. / Petersen, S. / Blaszczak, L.C. / Pulley, S.R. / Margolis, B.J. / Wishart, G.N. / Renson, B. / Hankotius, D. / Mohr, M. / Zechel, J.C. / Michael Kalbfleisch, J. / Dingess-Hammond, E.A. / Boelke, A. / Weichert, A.G.
External linksBioorg. Med. Chem. Lett. / PubMed:17239592
MethodsX-ray diffraction
Resolution2.1 Å
Structure data

PDB-2ogz:
Crystal structure of DPP-IV complexed with Lilly aryl ketone inhibitor
Method: X-RAY DIFFRACTION / Resolution: 2.1 Å

Chemicals

ChemComp-U1N:
4-[(3R)-3-{[2-(4-FLUOROPHENYL)-2-OXOETHYL]AMINO}BUTYL]BENZAMIDE

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsHYDROLASE / DIPEPTIDYL PEPTIDASE IV / CD26 / DPIV / DPP-IV / DPP4 / Serine Protease / inhibitor

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