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| Title | Thyroid Receptor Ligands. 6. A High Affinity "Direct Antagonist" Selective for the Thyroid Hormone Receptor. |
|---|---|
| Journal, issue, pages | J. Med. Chem., Vol. 49, Page 6635-, Year 2006 |
| Publish date | Aug 28, 2006 (structure data deposition date) |
Authors | Koehler, K. / Gordon, S. / Brandt, P. / Carlsson, B. / Backsbro-Saedi, A. / Apelqvist, T. / Agback, P. / Grover, G.J. / Nelson, W. / Grynfarb, M. ...Koehler, K. / Gordon, S. / Brandt, P. / Carlsson, B. / Backsbro-Saedi, A. / Apelqvist, T. / Agback, P. / Grover, G.J. / Nelson, W. / Grynfarb, M. / Farnegardh, M. / Rehnmark, S. / Malm, J. |
External links | J. Med. Chem. / PubMed:17154490 |
| Methods | X-ray diffraction |
| Resolution | 2.2 Å |
| Structure data | ![]() PDB-2j4a: |
| Chemicals | ![]() ChemComp-OEF: ![]() ChemComp-HOH: |
| Source |
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Keywords | RECEPTOR / NUCLEAR PROTEIN / DISEASE MUTATION / NUCLEAR RECEPTOR / ZINC / DEAFNESS / ZINC-FINGER / DNA-BINDING / TRANSCRIPTION REGULATION / TRANSCRIPTION / ALTERNATIVE SPLICING / LIGAND BINDING DOMAIN / POLYMORPHISM / METAL-BINDING |
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homo sapiens (human)
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