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-Structure paper
Title | Structural basis for the exceptional in vivo efficacy of bisphosphonate drugs. |
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Journal, issue, pages | Chemmedchem, Vol. 1, Page 267-273, Year 2006 |
Publish date | Dec 1, 2005 (structure data deposition date) |
![]() | Rondeau, J.M. / Bitsch, F. / Bourgier, E. / Geiser, M. / Hemmig, R. / Kroemer, M. / Lehmann, S. / Ramage, P. / Rieffel, S. / Strauss, A. ...Rondeau, J.M. / Bitsch, F. / Bourgier, E. / Geiser, M. / Hemmig, R. / Kroemer, M. / Lehmann, S. / Ramage, P. / Rieffel, S. / Strauss, A. / Green, J.R. / Jahnke, W. |
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Methods | X-ray diffraction |
Resolution | 1.94 - 2.6 Å |
Structure data | ![]() PDB-2f7m: ![]() PDB-2f89: ![]() PDB-2f8c: ![]() PDB-2f8z: ![]() PDB-2f92: ![]() PDB-2f94: ![]() PDB-2f9k: |
Chemicals | ![]() ChemComp-PO4: ![]() ChemComp-HOH: ![]() ChemComp-MN: ![]() ChemComp-210: ![]() ChemComp-MG: ![]() ChemComp-ZOL: ![]() ChemComp-IPE: ![]() ChemComp-ZN: ![]() ChemComp-AHD: ![]() ChemComp-BFQ: |
Source |
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![]() | TRANSFERASE / TRANSFERASE; ISOPRENE BIOSYNTHESIS; CHOLESTEROL BIOSYNTHESIS / MEVALONATE PATHWAY; ISOPRENE BIOSYNTHESIS; CHOLESTEROL BIOSYNTHESIS; BISPHOSPHONATE INHIBITOR / Mevalonate pathway / ; isoprene biosynthesis; cholesterol biosynthesis; bisphosphonate inhibitor |