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Structure paper

TitleLead optimization of methionine aminopeptidase-2 (MetAP2) inhibitors containing sulfonamides of 5,6-disubstituted anthranilic acids
Journal, issue, pagesBioorg. Med. Chem. Lett., Vol. 17, Page 2817-2822, Year 2007
Publish dateJan 30, 2007 (structure data deposition date)
AuthorsWang, G.T. / Mantei, R.A. / Kawai, M. / Tedrow, J.S. / Barnes, D.M. / Wang, J. / Zhang, Q. / Lou, P. / Garcia, L.A. / Bouska, J. ...Wang, G.T. / Mantei, R.A. / Kawai, M. / Tedrow, J.S. / Barnes, D.M. / Wang, J. / Zhang, Q. / Lou, P. / Garcia, L.A. / Bouska, J. / Yates, M. / Park, C. / Judge, R.A. / Lesniewski, R. / Sheppard, G.S. / Bell, R.L.
External linksBioorg. Med. Chem. Lett. / PubMed:17350258
MethodsX-ray diffraction
Resolution2.35 - 2.5 Å
Structure data

PDB-2ea2:
h-MetAP2 complexed with A773812
Method: X-RAY DIFFRACTION / Resolution: 2.5 Å

PDB-2ea4:
h-MetAP2 complexed with A797859
Method: X-RAY DIFFRACTION / Resolution: 2.35 Å

Chemicals

ChemComp-MN:
Unknown entry

ChemComp-F77:
3-ETHYL-6-{[(4-FLUOROPHENYL)SULFONYL]AMINO}-2-METHYLBENZOIC ACID

ChemComp-HOH:
WATER

ChemComp-F79:
2-(2-AMINOETHOXY)-3-ETHYL-6-{[(4-FLUOROPHENYL)SULFONYL]AMINO}BENZOIC ACID

Source
  • homo sapiens (human)
KeywordsHYDROLASE / Protein-ligand complex

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