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-Structure paper
Title | A 2.13 A Structure of E. coli Dihydrofolate Reductase Bound to a Novel Competitive Inhibitor Reveals a New Binding Surface Involving the M20 Loop Region |
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Journal, issue, pages | J. Med. Chem., Vol. 49, Page 6977-6986, Year 2006 |
Publish date | Aug 11, 2005 (structure data deposition date) |
![]() | Summerfield, R.L. / Daigle, D.M. / Mayer, S. / Mallik, D. / Hughes, D.W. / Jackson, S.G. / Sulek, M. / Organ, M.G. / Brown, E.D. / Junop, M.S. |
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Methods | X-ray diffraction |
Resolution | 2.13 - 2.68 Å |
Structure data | ![]() PDB-2ano: ![]() PDB-2anq: |
Chemicals | ![]() ChemComp-MN: ![]() ChemComp-NDP: ![]() ChemComp-817: ![]() ChemComp-HOH: ![]() ChemComp-C1A: |
Source |
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![]() | OXIDOREDUCTASE / DHFR / Protein inhibitor complex |