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-Structure paper
Title | Crystal structures of catalytic subunit of cAMP-dependent protein kinase in complex with isoquinolinesulfonyl protein kinase inhibitors H7, H8, and H89. Structural implications for selectivity. |
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Journal, issue, pages | J. Biol. Chem., Vol. 271, Page 26157-26164, Year 1996 |
Publish date | Jul 24, 1996 (structure data deposition date) |
![]() | Engh, R.A. / Girod, A. / Kinzel, V. / Huber, R. / Bossemeyer, D. |
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Methods | X-ray diffraction |
Resolution | 2.2 - 2.3 Å |
Structure data | ![]() PDB-1ydr: ![]() PDB-1yds: ![]() PDB-1ydt: |
Chemicals | ![]() ChemComp-IQP: ![]() ChemComp-HOH: ![]() ChemComp-IQS: ![]() ChemComp-IQB: |
Source |
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![]() | COMPLEX (PHOSPHOTRANSFERASE/INHIBITOR) / COMPLEX (PHOSPHOTRANSFERASE-INHIBITOR) / TRANSFERASE / CAMP / PHOSPHORYLATION / ISOQUINOLINE SULFONAMIDE / SERINE/THREONINE-PROTEIN KINASE / ATP-BINDING / COMPLEX (PHOSPHOTRANSFERASE-INHIBITOR) complex / TRANSFERASE/TRANSFERASE INHIBITOR / PHOSPHOTRANSFERASE / TRANSFERASE-TRANSFERASE INHIBITOR complex |