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-Structure paper
Title | Structural basis for the autoinhibition and STI-571 inhibition of c-Kit tyrosine kinase. |
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Journal, issue, pages | J. Biol. Chem., Vol. 279, Page 31655-31663, Year 2004 |
Publish date | Apr 28, 2004 (structure data deposition date) |
![]() | Mol, C.D. / Dougan, D.R. / Schneider, T.R. / Skene, R.J. / Kraus, M.L. / Scheibe, D.N. / Snell, G.P. / Zou, H. / Sang, B.C. / Wilson, K.P. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.6 - 1.9 Å |
Structure data | ![]() PDB-1t45: ![]() PDB-1t46: |
Chemicals | ![]() ChemComp-HOH: ![]() ChemComp-PO4: ![]() ChemComp-STI: |
Source |
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![]() | TRANSFERASE ACTIVATOR / KINASE / AUTOINHIBITION / INHIBITOR / STI-571 / Gleevec |