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Structure paper

TitleDesign of novel and selective inhibitors of urokinase-type plasminogen activator with improved pharmacokinetic properties for use as antimetastatic agents
Journal, issue, pagesJ. Biol. Chem., Vol. 279, Page 33613-33622, Year 2004
Publish dateFeb 12, 2004 (structure data deposition date)
AuthorsSchweinitz, A. / Steinmetzer, T. / Banke, I.J. / Arlt, M.J.E. / Stuerzebecher, A. / Schuster, O. / Geissler, A. / Giersiefen, H. / Zeslawska, E. / Jacob, U. ...Schweinitz, A. / Steinmetzer, T. / Banke, I.J. / Arlt, M.J.E. / Stuerzebecher, A. / Schuster, O. / Geissler, A. / Giersiefen, H. / Zeslawska, E. / Jacob, U. / Kruger, A. / Stuerzebecher, J.
External linksJ. Biol. Chem. / PubMed:15150279
MethodsX-ray diffraction
Resolution2 - 2.4 Å
Structure data

PDB-1sc8:
Urokinase Plasminogen Activator B-Chain-J435 Complex
Method: X-RAY DIFFRACTION / Resolution: 2.4 Å

PDB-1vj9:
Urokinase Plasminogen Activator B-Chain-JT464 Complex
Method: X-RAY DIFFRACTION / Resolution: 2.4 Å

PDB-1vja:
Urokinase Plasminogen Activator B-Chain-JT463 Complex
Method: X-RAY DIFFRACTION / Resolution: 2 Å

Chemicals

ChemComp-SO4:
SULFATE ION

ChemComp-2IN:
N-(BENZYLSULFONYL)SERYL-N~1~-{4-[AMINO(IMINO)METHYL]BENZYL}GLYCINAMIDE

ChemComp-HOH:
WATER

ChemComp-5IN:
N-(BENZYLSULFONYL)-L-SERYL-N~1~-{4-[AMINO(IMINO)METHYL]BENZYL}-O-BENZYL-L-SERINAMIDE

ChemComp-7IN:
N-(BENZYLSULFONYL)SERYL-N~1~-{4-[(Z)-AMINO(IMINO)METHYL]BENZYL}SERINAMIDE

Source
  • homo sapiens (human)
KeywordsHYDROLASE / UROKINASE / INHIBITOR / SERINE PROTEASE / HUMAN

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