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-Structure paper
Title | Identification of novel potent bicyclic peptide deformylase inhibitors |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 14, Page 1477-1481, Year 2004 |
Publish date | Jan 5, 2004 (structure data deposition date) |
![]() | Molteni, V. / He, X. / Nabakka, J. / Yang, K. / Kreusch, A. / Gordon, P. / Bursulaya, B. / Warner, I. / Shin, T. / Biorac, T. ...Molteni, V. / He, X. / Nabakka, J. / Yang, K. / Kreusch, A. / Gordon, P. / Bursulaya, B. / Warner, I. / Shin, T. / Biorac, T. / Ryder, N.S. / Goldberg, R. / Doughty, J. / He, Y. |
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Methods | X-ray diffraction |
Resolution | 1.95 Å |
Structure data | ![]() PDB-1s17: |
Chemicals | ![]() ChemComp-NI: ![]() ChemComp-GNR: ![]() ChemComp-GOL: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE / peptide deformylase inhibitor / rational drug design / antibiotic / protein-ligand complex |