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-Structure paper
Title | Potent, Selective Inhibitors of Protein Tyrosine Phosphatase 1B |
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Journal, issue, pages | BIOORG. MED. CHEM. LETT., Vol. 13, Page 1887-1890, Year 2003 |
Publish date | Feb 16, 2003 (structure data deposition date) |
Authors | Xin, Z. / Oost, T.K. / Abad-Zapatero, C. / Hajduk, P.J. / Pei, Z. / Szczepankiewicz, B.G. / Hutchins, C.W. / Ballaron, S.J. / Stashko, M.A. / Lubben, T. ...Xin, Z. / Oost, T.K. / Abad-Zapatero, C. / Hajduk, P.J. / Pei, Z. / Szczepankiewicz, B.G. / Hutchins, C.W. / Ballaron, S.J. / Stashko, M.A. / Lubben, T. / Trevillyan, J.M. / Jirousek, M.R. / Liu, G. |
External links | BIOORG. MED. CHEM. LETT. / PubMed:12749891 |
Methods | X-ray diffraction |
Resolution | 2.4 Å |
Structure data | PDB-1nz7: |
Chemicals | ChemComp-901: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / PROTEIN TYROSINE PHOSPHATASE FOLD / OXAMIC ACID INHIBITOR BOUND TO P-LOOP |