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-Structure paper
Title | Over-The-Barrier Transition State Analogues Provide New Chemistries for Inhibitor Design: The Case of Purine Nucleoside Phosphorylase |
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Journal, issue, pages | BIOCHEMISTRY, Vol. 42, Page 6057-6066, Year 2003 |
Publish date | Oct 28, 2002 (structure data deposition date) |
Authors | Lewandowicz, A. / Shi, W. / Evans, G.B. / Tyler, P.C. / Furneaux, R.H. / Basso, L.A. / Santos, D.S. / Almo, S.C. / Schramm, V.L. |
External links | BIOCHEMISTRY / PubMed:12755607 |
Methods | X-ray diffraction |
Resolution | 1.9 Å |
Structure data | PDB-1n3i: |
Chemicals | ChemComp-PO4: ChemComp-DIH: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / transition state complex / trimer / PNP |