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Title | An Ethylenamine Inhibitor Binds Tightly to Both Wild Type and Mutant HIV-1 Proteases. Structure and Energy Study |
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Journal, issue, pages | J. Med. Chem., Vol. 46, Page 1636-1644, Year 2003 |
Publish date | Jun 11, 2002 (structure data deposition date) |
![]() | Skalova, T. / Hasek, J. / Dohnalek, J. / Petrokova, H. / Buchtelova, E. / Duskova, J. / Soucek, M. / Majer, P. / Uhlikova, T. / Konvalinka, J. |
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Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | ![]() PDB-1lzq: |
Chemicals | ![]() ChemComp-0ZQ: ![]() ChemComp-BME: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / HIV / PEPTIDOMIMETIC / ethylenamine ISOSTERE / HYDROLASE-HYDROLASE INHIBITOR COMPLEX |