+Search query
-Structure paper
Title | Structure-based design of an osteoclast-selective, nonpeptide src homology 2 inhibitor with in vivo antiresorptive activity. |
---|---|
Journal, issue, pages | Proc. Natl. Acad. Sci. Usa, Vol. 97, Page 9373-9378, Year 2000 |
Publish date | Jul 17, 2000 (structure data deposition date) |
![]() | Shakespeare, W. / Yang, M. / Bohacek, R. / Cerasoli, F. / Stebbins, K. / Sundaramoorthi, R. / Azimioara, M. / Vu, C. / Pradeepan, S. / Metcalf, C. ...Shakespeare, W. / Yang, M. / Bohacek, R. / Cerasoli, F. / Stebbins, K. / Sundaramoorthi, R. / Azimioara, M. / Vu, C. / Pradeepan, S. / Metcalf, C. / Haraldson, C. / Merry, T. / Dalgarno, D. / Narula, S. / Hatada, M. / Lu, X. / van Schravendijk, M.R. / Adams, S. / Violette, S. / Smith, J. / Guan, W. / Bartlett, C. / Herson, J. / Iuliucci, J. / Weigele, M. / Sawyer, T. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.4 Å |
Structure data | ![]() PDB-1fbz: |
Chemicals | ![]() ChemComp-CC1: ![]() ChemComp-HOH: |
Source |
|
![]() | TRANSFERASE / SH2 DOMAIN / NONPEPTIDE INHIBITOR |