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-Structure paper
Title | Analyses of ligand binding in five endothiapepsin crystal complexes and their use in the design and evaluation of novel renin inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 36, Page 3809-3820, Year 1993 |
Publish date | Jul 27, 1994 (structure data deposition date) |
![]() | Lunney, E.A. / Hamilton, H.W. / Hodges, J.C. / Kaltenbronn, J.S. / Repine, J.T. / Badasso, M. / Cooper, J.B. / Dealwis, C. / Wallace, B.A. / Lowther, W.T. |
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Methods | X-ray diffraction |
Resolution | 1.9 Å |
Structure data | ![]() PDB-1epp: ![]() PDB-1epq: |
Chemicals | ![]() ChemComp-SO4: ![]() ChemComp-1Z1: ![]() ChemComp-HOH: ![]() ChemComp-0QF: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / HYDROLASE-HYDROLASE INHIBITOR COMPLEX / ACID PROTEINASE |