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-Structure paper
Title | Design of MKC-442 (emivirine) analogues with improved activity against drug-resistant HIV mutants. |
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Journal, issue, pages | J. Med. Chem., Vol. 42, Page 4500-4505, Year 1999 |
Publish date | Jul 21, 1999 (structure data deposition date) |
![]() | Hopkins, A.L. / Ren, J. / Tanaka, H. / Baba, M. / Okamato, M. / Stuart, D.I. / Stammers, D.K. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.5 Å |
Structure data | ![]() PDB-1c1b: ![]() PDB-1c1c: |
Chemicals | ![]() ChemComp-GCA: ![]() ChemComp-HOH: ![]() ChemComp-612: |
Source |
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![]() | TRANSFERASE / HIV-1 REVERSE TRANSCRIPTASE / AIDS / NON-NUCLEOSIDE INHIBITOR / DRUG DESIGN |