タイトル | PanDDA analysis -- Crystal Structure of PHIP in complex with Z198194396 synthetic derivative |
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ジャーナル・号・ページ | To Be Published |
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掲載日 | 2022年12月6日 (構造データの登録日) |
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著者 | Grosjean, H. / Aimon, A. / Hassell-Hart, S. / Bradshaw, W.J. / Krojer, T. / Talon, R. / Douangamath, A. / Koekemoer, L. / Biggin, P.C. / Spencer, J. / von Delft, F. |
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リンク | PubMedで検索 |
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手法 | X線回折 |
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解像度 | 1.3 - 1.55 Å |
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構造データ | PDB-8bw2: PanDDA analysis -- Crystal Structure of PHIP in complex with Z198194396 synthetic derivative 手法: X-RAY DIFFRACTION / 解像度: 1.35 Å PDB-8bw3: PanDDA analysis -- Crystal Structure of PHIP in complex with Z198194396 synthetic derivative 手法: X-RAY DIFFRACTION / 解像度: 1.3 Å PDB-8bw4: PanDDA analysis -- Crystal Structure of PHIP in complex with Z198194396 synthetic derivative 手法: X-RAY DIFFRACTION / 解像度: 1.55 Å |
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化合物 | ChemComp-Y3Y: (2R)-N-(2-methoxyethyl)-2-methyl-4-thiophen-2-ylcarbonyl-piperazine-1-carboxamide
ChemComp-Y3V: (2S)-N-(cyclopropylmethyl)-2-methyl-4-(1-methyl-1H-pyrrole-2-carbonyl)piperazine-1-carboxamide
ChemComp-Y3S: (2R)-4-(3-fluoranylthiophen-2-yl)carbonyl-N-(4-methoxyphenyl)-2-methyl-piperazine-1-carboxamide
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由来 | - homo sapiens (ヒト)
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キーワード | SIGNALING PROTEIN / brodomain / automated chemistry / reaction product |
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