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-Structure paper
タイトル | Development of allosteric and selective CDK2 inhibitors for contraception with negative cooperativity to cyclin binding. |
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ジャーナル・号・ページ | Nat Commun, Vol. 14, Page 3213-3213, Year 2023 |
掲載日 | 2021年8月19日 (構造データの登録日) |
![]() | Faber, E.B. / Sun, L. / Tang, J. / Roberts, E. / Ganeshkumar, S. / Wang, N. / Rasmussen, D. / Majumdar, A. / Hirsch, L.E. / John, K. ...Faber, E.B. / Sun, L. / Tang, J. / Roberts, E. / Ganeshkumar, S. / Wang, N. / Rasmussen, D. / Majumdar, A. / Hirsch, L.E. / John, K. / Yang, A. / Khalid, H. / Hawkinson, J.E. / Levinson, N.M. / Chennathukuzhi, V. / Harki, D.A. / Schonbrunn, E. / Georg, G.I. |
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手法 | X線回折 |
解像度 | 1.5 - 2 Å |
構造データ | ![]() PDB-7rwf: ![]() PDB-7s84: ![]() PDB-8fow: ![]() PDB-8fp0: ![]() PDB-8fp5: |
化合物 | ![]() ChemComp-EDO: ![]() ChemComp-7TW: ![]() ChemComp-HOH: ![]() ChemComp-8IL: ![]() ChemComp-1QK: ![]() ChemComp-RRC: ![]() ChemComp-ATP: ![]() ChemComp-MG: |
由来 |
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![]() | CELL CYCLE / Serine/threonine-protein kinase DNA repair Meiosis allosteric inhibitor drug development / allosteric inhibitor / drug development / kinase / Transferase / allosteric / inhibitor |