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-Structure paper
タイトル | Pan-SMARCA/PB1 Bromodomain Inhibitors and Their Role in Regulating Adipogenesis. |
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ジャーナル・号・ページ | J. Med. Chem., Vol. 63, Page 14680-14699, Year 2020 |
掲載日 | 2020年7月6日 (構造データの登録日) |
![]() | Wanior, M. / Preuss, F. / Ni, X. / Kramer, A. / Mathea, S. / Gobel, T. / Heidenreich, D. / Simonyi, S. / Kahnt, A.S. / Joerger, A.C. / Knapp, S. |
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手法 | X線回折 |
解像度 | 1.14 - 2.02 Å |
構造データ | ![]() PDB-6zn6: ![]() PDB-6znv: ![]() PDB-6zs2: ![]() PDB-6zs3: ![]() PDB-6zs4: |
化合物 | ![]() ChemComp-QMT: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-QMW: ![]() ChemComp-ZN: ![]() ChemComp-CL: ![]() ChemComp-ACT: ![]() ChemComp-FX5: ![]() ChemComp-QP8: |
由来 |
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![]() | PROTEIN BINDING / Bromodomain Inhibitor Epigenetics / GENE REGULATION / BROMODOMAIN / ATP-DEPENDENT HELICASE SMARCA4 / BRG1-ASSOCIATED FACTOR 190A / BAF190A / MITOTIC GROWTH AND TRANSCRIPTION ACTIVATOR / PROTEIN BRG-1 / PROTEIN BRAHMA HOMOLOG 1 / SNF2-BETA / SWI/SNF-RELATED MATRIX-ASSOCIATED ACTIN-DEPENDENT REGULATOR OF CHROMATIN SUBFAMILY A MEMBER 4 / STRUCTURAL GENOMICS CONSORTIUM / SGC / TRANSCRIPTION / COMPLEX / SMALL MOLECULE |