Halogen Atoms in the Protein-Ligand System. Structural and Thermodynamic Studies of the Binding of Bromobenzotriazoles by the Catalytic Subunit of Human Protein Kinase CK2.
PDB-6tll: HUMAN CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE ATP-COMPETITIVE INHIBITOR 4,5,6,7-TETRABROMOBENZOTRIAZOLE (tBBT) 手法: X-RAY DIFFRACTION / 解像度: 1.88 Å
PDB-6tlo: HUMAN CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE ATP-COMPETITIVE INHIBITOR 4,5,6-TRIBROMOBENZOTRIAZOLE 手法: X-RAY DIFFRACTION / 解像度: 1.69 Å
PDB-6tlp: HUMAN CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE ATP-COMPETITIVE INHIBITOR 5,6-DIBROMOBENZOTRIAZOLE 手法: X-RAY DIFFRACTION / 解像度: 1.93 Å
PDB-6tlr: HUMAN CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE ATP-COMPETITIVE INHIBITOR 4,7-DIBROMOBENZOTRIAZOLE 手法: X-RAY DIFFRACTION / 解像度: 1.64 Å
PDB-6tls: HUMAN CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE ATP-COMPETITIVE INHIBITOR 4,6-DIBROMOBENZOTRIAZOLE 手法: X-RAY DIFFRACTION / 解像度: 1.46 Å
PDB-6tlu: HUMAN CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE ATP-COMPETITIVE INHIBITOR 4,5-DIBROMOBENZOTRIAZOLE 手法: X-RAY DIFFRACTION / 解像度: 1.81 Å
PDB-6tlv: HUMAN CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE ATP-COMPETITIVE INHIBITOR 5-BROMOBENZOTRIAZOLE 手法: X-RAY DIFFRACTION / 解像度: 1.67 Å
PDB-6tlw: HUMAN CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE ATP-COMPETITIVE INHIBITOR 4-BROMOBENZOTRIAZOLE 手法: X-RAY DIFFRACTION / 解像度: 1.73 Å