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-Structure paper
タイトル | Selective targeting of BD1 and BD2 of the BET proteins in cancer and immunoinflammation. |
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ジャーナル・号・ページ | Science, Vol. 368, Page 387-394, Year 2020 |
掲載日 | 2019年9月22日 (構造データの登録日) |
![]() | Gilan, O. / Rioja, I. / Knezevic, K. / Bell, M.J. / Yeung, M.M. / Harker, N.R. / Lam, E.Y.N. / Chung, C.W. / Bamborough, P. / Petretich, M. ...Gilan, O. / Rioja, I. / Knezevic, K. / Bell, M.J. / Yeung, M.M. / Harker, N.R. / Lam, E.Y.N. / Chung, C.W. / Bamborough, P. / Petretich, M. / Urh, M. / Atkinson, S.J. / Bassil, A.K. / Roberts, E.J. / Vassiliadis, D. / Burr, M.L. / Preston, A.G.S. / Wellaway, C. / Werner, T. / Gray, J.R. / Michon, A.M. / Gobbetti, T. / Kumar, V. / Soden, P.E. / Haynes, A. / Vappiani, J. / Tough, D.F. / Taylor, S. / Dawson, S.J. / Bantscheff, M. / Lindon, M. / Drewes, G. / Demont, E.H. / Daniels, D.L. / Grandi, P. / Prinjha, R.K. / Dawson, M.A. |
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手法 | X線回折 |
解像度 | 1.28 - 1.604 Å |
構造データ | ![]() PDB-6swn: ![]() PDB-6swo: ![]() PDB-6swp: ![]() PDB-6swq: |
化合物 | ![]() ChemComp-GLU: ![]() ChemComp-LWB: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-LW5: |
由来 |
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![]() | TRANSCRIPTION / INHIBITOR / HISTONE / EPIGENETIC READER / BROMODOMAIN / BRD4 / BROMODOMAIN CONTAINING PROTEIN 4 / ANTAGONIST / BRD2 / BROMODOMAIN CONTAINING PROTEIN 2 / BROMODOMAIN CONTAINING PROTEIN4 |